Inventors:
- Princeton NJ, US
Collin Chan - New York NY, US
Joerg Deerberg - Columbus NJ, US
Nathan R. Domagalski - Niantic CT, US
Martin D. Eastgate - Titusville NJ, US
Yu Fan - Highland Park NJ, US
Michael David Bengt Fenster - New York NY, US
Robert V. Forest - Hillsborough NJ, US
Rebecca A. Green - Metuchen NJ, US
Matthew R. Hickey - Yardley PA, US
Nathaniel David Kopp - Newtown PA, US
Thomas E. La Cruz - Flemington NJ, US
Kathleen Lauser - Minneapolis MN, US
Hong Geun Lee - Seoul, KR
David K. Leahy - Hightstown NJ, US
Helen Y. Luo - San Francisco CA, US
Thomas M. Razler - Yardley PA, US
Scott A. Savage - Yardley PA, US
Chris Sfouggatakis - Staten Island NY, US
Maxime C.D. Soumeillant - Princeton NJ, US
Serge Zaretsky - Fords NJ, US
Bin Zheng - Kendall Park NJ, US
Ye Zhu - Singapore, SG
International Classification:
C07D 487/04
Abstract:
The invention generally relates to an improved process for the preparation of N-((1R,2S,5R)-5-(tert-butylamino)-2-((S)-3-(7-tert-butylpyrazolo[1,5-a][1,3,5]triazin-4-ylamino)-2-oxopyrrolidin-1-yl)cyclohexyl)acetamide,