US Patent:
20150210697, Jul 30, 2015
Inventors:
- Princeton NJ, US
Brian E. Fink - Yardley PA, US
Walter Lewis Johnson - Waterbury CT, US
Amy C. Hart - Ewing NJ, US
Liqi He - Furlong PA, US
Tram N. Huynh - Pennington NJ, US
Jennifer Inghrim - Plainsboro NJ, US
Harold Mastalerz - Guilford CT, US
Xiaopeng Sang - Glastonbury CT, US
Christine M. Tarby - Lawrenceville NJ, US
Honghe Wan - Pennington NJ, US
Wayne Vaccaro - Yardley PA, US
Guifen Zhang - Wallingford CT, US
Yufen Zhao - Pennington NJ, US
Kurt Zimmermann - Durham CT, US
Yong Zhang - Princeton Junction NJ, US
Libing Chen - Newtown PA, US
Bin Chen - Pennington NJ, US
John S. Tokarski - Princeton NJ, US
Ashvinikumar V. Gavai - Princeton Junction NJ, US
International Classification:
C07D 487/04
C07F 7/18
C07D 487/10
C07D 487/08
C07D 471/10
Abstract:
The invention provides compounds of Formula (I) and pharmaceutically acceptable salts thereof. The Formula (I) imidazotriazines inhibit protein kinase activity thereby making them useful as anticancer agents.