Inventors:
Donald B Borders - Suffern NY
William V Curran - Pearl River NY
Amedeo A Fantini - New City NY
Noreen D Francis - Harriman NY
Howard Jarolmen - Upper Saddle River NJ
Richard A Leese - Suffern NY
Assignee:
Micrologix Biotech Inc. - Vancouver
International Classification:
A61K 3812
US Classification:
514 11, 435 681, 435 713, 530317
Abstract:
The present invention provides a laspartomycin core peptide, a laspartomycin core peptide derivative, a antimicrobial laspartomycin derivative, a method for making laspartomycin core peptides, methods for making laspartomycin core peptide derivatives, methods for making antimicrobial laspartomycin derivatives, pharmaceutical compositions of antimicrobial laspartomycin derivatives, methods of inhibiting microbial growth and methods for treating and/or preventing microbial infections in a subject.